Tuesday, July 16, 2024

Cardiovascular Diseases: How Best to Manage Them?

Cardiovascular Diseases


ju-boo lim 

The most common cardiovascular diseases (CVDs) seen today include coronary artery disease (CAD), hypertension (high blood pressure), heart failure, arrhythmias, and stroke. Managing these conditions without drugs involves lifestyle modifications and preventive measures that can significantly reduce the risk and progression of CVDs.

These include coronary artery disease (CAD) caused by atherosclerosis (plaque buildup in arteries). Patients normally complain of chest pain (angina), shortness of breath, heart attack

However, before they get to CAD, the most common we see would-be hypertension (high blood pressure). Many people think and blame hypertension caused by genetic factors, and they give excuses that they cannot do anything about this. But I think hypertension is mainly caused by unhealthy eating such as excessive salt intake, lack of exercise, and obesity. Often hypertension is asymptomatic but can lead to complications like stroke and heart attack. If we can eat healthily, we can override the expression of genetics if we think that hypertension is carried down by our parents and there is nothing, we can do about this? Is this really true?  Blame our lifestyle and eating habits first, not our parents who have nothing to do with the ways we live our lives.

CVD may lead to heart failure caused by CAD, hypertension, cardiomyopathy, heart valve disease. The symptoms presented are shortness of breath, fatigue, swollen legs, rapid heartbeat.

Another CVS is arrhythmia caused by CAD, heart failure, electrolyte imbalances and medications which I shall discuss shortly.

In arrhythmia or irregular heartbeats, patient would complain of palpitations, dizziness, fainting, shortness of breath

One of the most common of CVD is cerebrovascular accident (CVA), brain attack) or stroke. This is caused by a blockage or rupture of blood vessels in the brain. In a stroke there is a sudden weakness or numbness, confusion, trouble speaking, severe headache

What would be the best methods to manage and prevent cardiovascular diseases without drugs

Let’s have a look together.

First, is to adopt a health-protective diet such as a Mediterranean diet rich in fruits, vegetables, whole grains, lean proteins, and healthy fats (e.g., olive oil, nuts). Nutrition in the prevention of almost all diseases is exceedingly important not just for cardiovascular diseases or metabolic and endocrine diseases like diabetes mellitus. This diet is associated with lower risks of heart disease. More important is to reduce sodium intake.  Limiting salt helps manage blood pressure.

Limit also the consumption of saturated and trans fats such as animal fats and margarine. Reducing these fats lowers cholesterol levels. White, refined sugar is very deadly, according to Professor John Yudkin who was the Chair of Nutrition at the University of London.  Sugar (sucrose) is the primary cause of coronary heart disease, and I strongly support this theory.

In order to prevent CAD, it is also important to increase fibre intake by consuming whole grains, fruits, and vegetables. Intake of these foods help maintain a healthy heart.

Regular physical activity such as aerobic exercise like walking, moderate running, cycling, or swimming for at least 150 minutes per week. Consider also strength training, muscle-strengthening activities at least twice a week or flexibility and balance exercises to include yoga or tai chi to improve overall physical health.

But importantly is weight management to prevent overweight and obesity. Maintaining a healthy weight reduces the strain on the heart and lowers the risk of hypertension, CAD, and diabetes.

We need also to consider a balanced caloric intake to ensure that calorie intake matches energy expenditure to prevent weight gain.

One of the other causes of CAD is smoking besides the risk of developing lung cancer. Avoid tobacco since smoking is a major risk factor for CVD. Quitting smoking reduces the risk significantly.  By this, I mean also to avoid second hand smoke as exposure to second-hand smoke in crowded places where people smoke. Exposure to second hand smoke also increases the risk of heart disease.

If you drink, moderate drinking is strongly advisable. Alcohol consumption should be in moderation (up to one drink per day for women and up to two drinks per day for men.

Another factor to prevent CAD is stress management. Practicing relaxation techniques such as meditation, deep breathing exercises, and mindfulness can reduce stress. Regular exercise too helps manage stress and improve mental health.

Ensuring you have adequate sleep (7-9 hours per night) is crucial for heart health.

Regular checks on blood pressure are preventive.  Regular monitoring to ensure blood pressure remains within a healthy range. Regular testing for blood cholesterol may be useful to maintain healthy cholesterol levels although there is a lot of disagreement if high cholesterol levels is the cause of cardiovascular disease

Does Cholesterol Cause Heart Disease?

https://scientificlogic.blogspot.com/search?q=cholesterol+does+not+cause+heart+disease

But I think diabetes screening would be more useful as early detection and management of diabetes reduce the risk of CVD.

But what are the larger scale prevention strategies? I believe in education.  Educate and raise awareness. By this I mean understanding the risk factors and symptoms of CVDs can lead to early intervention and lifestyle changes.

We can also have Community Programs by participating in community health programs that promote physical activity and healthy eating. We can also have support networks by joining support groups for smoking cessation, weight loss, or stress management can provide motivation and resources.

We can have public policies. We can advocate for policies that promote healthy environments, such as smoke-free zones, availability of healthy food options, and safe spaces for physical activities.

By adopting these lifestyle changes and preventive measures, individuals can significantly reduce their risk of developing cardiovascular diseases and manage existing conditions more effectively without relying solely on medications. Prevention is always better than cure.

But what if CVD has set in and medication is needed.

Let us now look at the treatment aspect using drugs and medication that I strongly would try to avoid. But let us say drugs are now needed to manage cases of CVD. Let’s have a short discussion about the use of various vascular drugs.

Treating cardiovascular diseases involves a range of medications, each targeting different aspects of heart and blood vessel function.  The various kinds of drugs used, including their dosages, advantages, disadvantages, and effectiveness.

There are antihypertensives drugs to manage hypertension. Examples of these would include:

Angiotensin-Converting Enzyme (ACE) Inhibitors such as Lisinopril, Enalapril, Ramipril. The dosage for Lisinopril is 10-40 mg once daily, Enalapril is given at 5-40 mg once daily or divided doses and Ramipril titrated at 2.5-20 mg once daily

The advantages is, it is effective in lowering blood pressure, improving heart function, and reducing the risk of stroke and heart attack. The disadvantages with these drugs are they can cause cough, elevated blood potassium levels, low blood pressure, and kidney dysfunction. However, their effectiveness is high, particularly in patients with heart failure or diabetes.

Then there are Angiotensin II Receptor Blockers (ARBs) such as the popular Losartan, Valsartan, or combined with a diuretic such as hydrochlorothiazide as in Co-Diovan used to treat high blood pressure. Another example of antihypertensive is Telmisartan The dosage for Losartan is 50-100 mg once daily, Valsartan is 80-320 mg once daily and Telmisartan (rarely used) is 20-80 mg once daily.

The advantage with this medication is, they can lower blood pressure and risk of heart failure, with fewer side effects than ACE inhibitors. The disadvantages are, they may cause dizziness, elevated blood potassium, and kidney dysfunction. The effectiveness is similar to ACE inhibitors, often used as an alternative.

We also have beta-blockers such as Metoprolol, Atenolol, Carvedilol. The dosages normally prescribed are Metoprolol at 50-200 mg once daily, Atenolol given at 25-100 mg once daily and Carvedilol given at 12.5-50 mg twice daily

The advantages with these drugs are they reduce heart rate, blood pressure, and risk of heart attacks; improve survival in heart failure patients. The disadvantages are they can cause fatigue, cold extremities, depression, and sexual dysfunction. Their effectiveness is high, especially post-heart attack and in heart failure management.

Cholesterol-lowering drugs are the statins groups. These include (examples) Atorvastatin, Simvastatin, Rosuvastatin The dosage for Atorvastatin is 10-80 mg once daily, Simvastatin given at 10-40 mg once daily and Rosuvastatin at 5-40 mg once daily. Lipitor is another commonly used statin. The dosage for Lipitor is between 10 – 20 mg once a day preferably at night when cholesterol is mostly synthesized by the liver.

These statins significantly lower LDL cholesterol, reduce risk of heart attack and stroke.

The disadvantage with statins is, they can cause muscle pain, liver enzyme elevation, and increased blood sugar levels. Their clinical efficacies are very high in preventing cardiovascular events.

Sometimes Ezetimibe is also being prescribed elsewhere. The dosage is 10 mg once daily This drug also reduces LDL cholesterol by inhibiting absorption in the intestines.

However its disadvantage is, it can cause gastrointestinal issues and muscle pain. It is often used in combination with statins for better effectiveness. I think most doctors would not bother to monitor the liver enzyme levels when they prescribe all these statins because these statins can damage the liver. I would strongly advise conducting liver function tests when we use statins for at least the first few months, and perhaps at 6 months intervals after that. We must not assume using all these drugs are safe without monitoring. All drugs are chemicals and are poisons and they can cause acute reactions or accumulative poisoning especially used for chronic disorders over long term.   

Next, we come to the antiplatelet agents. The most common is aspirin given at 75-325 mg once daily. However, there are 100 mg presentation tablets that can be used especially at night after dinner.

Aspirin can reduce the risk of heart attack and stroke by preventing blood clots. However, the disadvantage with aspirin is, it can cause gastrointestinal bleeding and ulcers. Nevertheless, aspirin effectiveness ranges from moderate to high, widely used for secondary prevention.

Another antiplatelet agent is Clopidogrel. This is prescribed for the prevention of blood clots, often used in patients who can't take aspirin. Its disadvantages, like aspirin, the risk of bleeding, gastrointestinal issues. Nevertheless, its effectiveness is high, especially in combination with aspirin for certain conditions. The dosage for Clopidogrel is 75 mg once daily. This can also be prescribed to prevent blood clots, often used in patients who can't take aspirin.  But there is also the risk of bleeding and gastrointestinal issues.

Next, are the anticoagulants used for CVD. An example is warfarin. The dosage is individualized based on INR (International Normalized Ratio) monitoring, Warfarin advantages are effective in preventing blood clots in conditions like atrial fibrillation and after certain surgeries. But its disadvantages are, warfarin requires regular blood monitoring, risk of bleeding, interactions with foods and other medications. In short, warfarin effectiveness is high, but requires careful management.

Examples of other direct oral anticoagulants (DOACs) are Apixaban, Rivaroxaban, and Dabigatran The dosages for Apixaban is 2.5-5 mg twice daily, Rivaroxaban is 10-20 mg once daily and for Dabigatran it is given at 150 mg twice daily. The advantage with these three DOACs is, no regular blood monitoring is needed, fewer food and drug interactions. But their disadvantages are, the risk of bleeding which is not easily reversible in case of emergency. But its effectiveness is high, often preferred over warfarin for ease of use.

But I think diuretics such as thiazide diuretics should be considered as the first line of choice in the management of CVD especially for hypertension.

Examples of water-throwing drugs are hydrochlorothiazide and chlorthalidone

The dosages normally given for hydrochlorothiazide is 12.5-50 mg once daily and for chlorthalidone is, 12.5-25 mg once daily

The advantages with diuretics are their effectiveness in lowering blood pressure and reducing fluid retention. The disadvantage with diuretics is, they can cause electrolyte imbalances, dehydration, and increased blood sugar. Nevertheless, the effectiveness with diuretics is high, and this should be first-line treatment for hypertension.

We can also consider using loop diuretics Furosemide prescribed at 20 -80 mg once or twice a day, and Bumetanide given at 0.5 – 2 mg once or twice a day are two examples with loop diuretics.

These two are powerful diuretics, effective in reducing oedema and fluid overload in heart failure. Like all drugs there are disadvantages. With diuretics there is always the risk of electrolyte imbalances, dehydration, kidney dysfunction. Despite that, its clinical efficacy is very high in managing heart failure symptoms.

Next, we also have the calcium channel blockers (CCB). Examples of CCB are Amlodipine, Diltiazem, Verapamil where Amlodipine is prescribed at 5-10 mg once daily, Diltiazem given at 120-360 mg once daily and Verapamil at 80-120 mg three times daily or extended-release formulations

These agents lower blood pressure, reduce chest pain (angina), and control heart rate.

But they can cause swelling, constipation, dizziness, and heart rate irregularities.

Their clinical efficacy is quite high for hypertension and angina, moderate for heart rate control.

There are also the nitrates such as nitro-glycerine, and Isosorbide Mononitrate

Nitro-glycerine is normally given at 0.3-0.6 mg sublingually as needed for chest pain whereas Isosorbide Mononitrate is prescribed at 20-60 mg once or twice daily

These nitrates relieve chest pain (angina), improve blood flow to the heart. Unfortunately, they can cause headaches, dizziness, low blood pressure, and tolerance with long-term use. Efficacy for nitrates is high for angina relief, especially in acute settings.

I may say, the effectiveness of these medications varies based on individual patient conditions and comorbidities. A physician typically customizes the treatment plan to achieve the best outcomes, balancing benefits and potential side effects. Regular monitoring and follow-ups are crucial to ensure optimal effectiveness and safety of the prescribed regimen. We normally consider benefit and risk ratios when we use risky drugs.

But once again, I would strongly like to emphasize on prevention rather than using all these drugs to solve a problem.  I don’t believe using drugs is the right way to acquire health. All these drugs should be used last.

Prevention for most diseases, especially for modern chronic lifestyle diseases also known as non-communicable diseases (NCDs), are typically caused by a combination of genetic, physiological, environmental, and behavioural factors that are best treated by lifestyle changes.  These diseases are long-lasting and often progress slowly. The main chronic lifestyle diseases include:

Cardiovascular Diseases like coronary artery disease, hypertension (high blood pressure), stroke, congestive heart failure, diabetes mellitus. Type 2 diabetes and prediabetes, chronic respiratory diseases such as chronic obstructive pulmonary disease (COPD) like chronic bronchitis, emphysema, asthma should be treated by addressing their root causes as first line management.

Not just CVD only but also cancers like lung, breast, colorectal, prostate cancers, and even skin cancer (melanoma and non-melanoma). Other lifestyle diseases are obesity, metabolic syndrome, chronic kidney disease, liver diseases such as non-alcoholic fatty liver disease (NAFLD), cirrhosis, arthritis like osteoporosis, osteoarthritis, rheumatoid arthritis, mental health disorders such as depression, anxiety disorders, not forgetting neurological disorders (examples are Alzheimer's disease and Parkinson's disease), and gastrointestinal diseases (examples are, irritable bowel syndrome (IBS), inflammatory bowel disease (IBD), including Crohn's disease and ulcerative colitis).

These diseases are often influenced by lifestyle factors such as diet, physical activity, tobacco use, and alcohol consumption. Prevention and management typically involve lifestyle changes, such as adopting a healthy diet, regular physical activity, maintaining a healthy weight, avoiding tobacco use, and limiting alcohol consumption.

 Even if a patient is on medication for some form of cardiovascular disease, that does not mean he cannot change his dietary lifestyles or engage in some light physical activities, such as tai chi and qigong, indulges in stress management and mediation, perhaps not strenuous exercise if he suffers from or has a history of coronary heart disease where there may be a risk here:

https://scientificlogic.blogspot.com/2024/07/do-you-think-exercise-and-jogging-are.html

He may even benefit from these activities even if he suffers from heart block.  

Heart block does not mean the coronary vessels of the heart are blocked by fatty plaque buildup. That is arteriosclerosis, not heart block. Heart block, also known as atrioventricular (AV) block, is a condition where the electrical signals that control the heartbeat are partially or completely blocked as they travel from the atria (upper chambers of the heart) to the ventricles (lower chambers). This disruption can cause the heart to beat irregularly and more slowly than normal. Heart block is classified into three main degrees based on the severity of the block.

First-degree heart block is the mildest form where electrical signals are slowed but still reach the ventricles. The ECG characteristics show prolonged PR intervals (greater than 0.20 seconds) without missed beats. Often asymptomatic; typically discovered incidentally during an ECG.

In the second-degree heart block some electrical signals from the atria fail to reach the ventricles. In the second-degree heart block, there are two types. There is the Mobitz Type I (Wenckebach) in which the ECG characteristics show progressive lengthening of the PR interval until a beat is dropped. The patient is often asymptomatic but may cause dizziness or palpitations. In the Mobitz Type II, the ECG shows sudden dropped beats without a change in PR interval length. More likely to cause symptoms such as dizziness, syncope (fainting), and can progress to complete heart block.

Third-degree (complete) heart block shows no electrical signals reach the ventricles from the atria. The atria and ventricles beat independently of each other. The ECG shows no relationship between P waves and QRS complexes; atrial rate is faster than the ventricular rate. This can cause severe symptoms such as fatigue, dizziness, syncope, and can be life-threatening.

Dietary changes, physical activity, control of body weight, stress reduction themselves can bring about tremendous changes for the better to his existing cardiovascular problems. It may not be surprising that he may no longer need any more medication if he takes the trouble to institute all these health promoting changes. Take heed, the body has amazing ability to heal itself if not continuously injured by harmful living and destructive exposures such as consumption of harmful foods, excessive eating, contacts with chemicals, intake of unnecessary drugs and medication, exposure to infective agents, radiation, free radicals, smoking, constant trauma and injuries from external and internal stress, etc. Once these injurious agents are removed, the body begins to repair itself from the damages especially if we can stimulate, massage, needle, coax, nourish and rest it. By and by the body restore itself, till finally we may no longer need any of those medication that do not cure or heal anything  

As a former senior medical researcher and a clinician, I would place prevention of all these NCDs first rather than trying to look for a “cure” using all these drugs that are actually chemicals that the body tries to break down and throw away into the urine.

I am not very happy and comfortable using all these chemicals under the hidden and glorified name called “medicine” to “cure” most of our modern lifestyle diseases.   

I hope my essays and efforts here and elsewhere are useful and educational for everyone, including medical doctors who are more interested in prescribing drugs and promoting all these chemical pharmaceuticals the easy and short-cut way than addressing the root causes and educating the patient.

 

References:

For further reading on medicines and drugs here are a few:

1.      The Dilemma Between the Doctor, the Patient and the Drugs They Take

https://scientificlogic.blogspot.com/search?q=pharmacology

2.      Ancient Medicine and Modern Medicine: My Personal Experience

Scientific Logic: Search results for history of medicine

3.      Synthetic Drugs vs Botanical and Herbal Medicines. Which is Better?

https://scientificlogic.blogspot.com/2024/05/my-brother-in-law-ong-geok-soo-senior.html

4.      All On Drugs. How Do They Work? Are They Safe?

 https://scientificlogic.blogspot.com/search?q=emergency+drugs

Here are some other recent studies and reviews on the clinical efficacy and dosage of various cardiovascular drugs:

1.  Statins (Rosuvastatin vs. Atorvastatin): The LODESTAR trial conducted in South Korea compared the efficacy of rosuvastatin and atorvastatin in adults with coronary artery disease. Participants were randomized to either a treat-to-target strategy with titrated statin intensity to achieve LDL cholesterol levels of 1.3-1.8 mmol/L or a high-intensity statin strategy irrespective of LDL levels. The trial demonstrated that both statins effectively managed dyslipidemia, with particular emphasis on adherence to the assigned statin type throughout the follow-up period (BMJ).

2.  Sacubitril/Valsartan (Entresto): Sacubitril/valsartan has shown significant clinical benefits in heart failure patients compared to valsartan alone. This combined therapy not only improves heart failure symptoms but also reduces hospitalizations and cardiovascular death. The shift from monotherapy to combination therapy has marked an important advancement in cardiovascular pharmacotherapy (Frontiers)

3.  Semaglutide (Wegovy): The SELECT trial investigated the cardiovascular benefits of semaglutide 2.4 mg in overweight or obese individuals without diabetes but with established cardiovascular disease. The study found a 20% reduction in major adverse cardiovascular events (MACE) compared to placebo. Semaglutide's safety profile was consistent with previous trials, highlighting its potential to change obesity treatment paradigms by reducing cardiovascular risks (Novo Nordisk).

These studies illustrate ongoing efforts to optimize cardiovascular drug therapies, emphasizing tailored treatment strategies to improve patient outcomes. For more detailed information, you can access the full articles and reviews in the respective medical journals and publications.

Take Care!

Jb

 

 

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